Synthesis of prenylated benzaldehydes and their use in the synthesis of analogues of licochalconeA (Record no. 43401)
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| 000 -LEADER | |
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| fixed length control field | 01586nam a2200217Ia 4500 |
| 003 - CONTROL NUMBER IDENTIFIER | |
| control field | MX-MdCICY |
| 005 - DATE AND TIME OF LATEST TRANSACTION | |
| control field | 20250625124733.0 |
| 040 ## - CATALOGING SOURCE | |
| Transcribing agency | CICY |
| 090 ## - LOCALLY ASSIGNED LC-TYPE CALL NUMBER (OCLC); LOCAL CALL NUMBER (RLIN) | |
| Classification number (OCLC) (R) ; Classification number, CALL (RLIN) (NR) | B-9143 |
| 008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION | |
| fixed length control field | 250602s9999 xx |||||s2 |||| ||und|d |
| 245 10 - TITLE STATEMENT | |
| Title | Synthesis of prenylated benzaldehydes and their use in the synthesis of analogues of licochalconeA |
| 490 0# - SERIES STATEMENT | |
| Volume/sequential designation | European Journal of Medicinal Chemistry, 39(11), 2004 |
| 520 3# - SUMMARY, ETC. | |
| Summary, etc. | In this paper, a general applicable synthesis of prenylated aromatic compounds exemplified by prenylated benzaldehydes starting from readily available acetophenones is described. The synthesized benzaldehydes are used to prepare a number of novel analogues of Licochalcone A, a known antibacterial compound, and for the exploration of the pharmacophoric elements that are essential for the antibacterial activity. It is shown that the hydroxyl group in the A ring is essential for the activity and that the hydroxyl group in the B ring has no influence on the antibacterial effect of Licochalcone A. Furthermore, it is shown that the prenyl group at the position 5 f the B ring also has a dominating influence on the activity. This aliphatic group can be replaced by other lipophilic long chained substituents in order to maintain the activity. |
| 700 12 - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Kromann, H. |
| 700 12 - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Larsen, M. |
| 700 12 - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Boesen, T. |
| 700 12 - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Schønning, K. |
| 700 12 - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Nielsen, S.F. |
| 856 40 - ELECTRONIC LOCATION AND ACCESS | |
| Uniform Resource Identifier | <a href="https://drive.google.com/file/d/1rYcBZ0aWL7DjHRkMzOxu7UJy02Q2EOFv/view?usp=drivesdk">https://drive.google.com/file/d/1rYcBZ0aWL7DjHRkMzOxu7UJy02Q2EOFv/view?usp=drivesdk</a> |
| Public note | Para ver el documento ingresa a Google con tu cuenta: @cicy.edu.mx |
| 942 ## - ADDED ENTRY ELEMENTS (KOHA) | |
| Source of classification or shelving scheme | Clasificación local |
| Koha item type | Documentos solicitados |
| Lost status | Source of classification or shelving scheme | Damaged status | Not for loan | Collection | Home library | Current library | Shelving location | Date acquired | Total checkouts | Full call number | Date last seen | Price effective from | Koha item type |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Clasificación local | Ref1 | CICY | CICY | Documento préstamo interbibliotecario | 25.06.2025 | B-9143 | 25.06.2025 | 25.06.2025 | Documentos solicitados |
