Salt selection for basic drugs (Record no. 49135)
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| 000 -LEADER | |
|---|---|
| fixed length control field | 01524nam a2200193Ia 4500 |
| 003 - CONTROL NUMBER IDENTIFIER | |
| control field | MX-MdCICY |
| 005 - DATE AND TIME OF LATEST TRANSACTION | |
| control field | 20250625153951.0 |
| 040 ## - CATALOGING SOURCE | |
| Transcribing agency | CICY |
| 090 ## - LOCALLY ASSIGNED LC-TYPE CALL NUMBER (OCLC); LOCAL CALL NUMBER (RLIN) | |
| Classification number (OCLC) (R) ; Classification number, CALL (RLIN) (NR) | B-14951 |
| 008 - FIXED-LENGTH DATA ELEMENTS--GENERAL INFORMATION | |
| fixed length control field | 250602s9999 xx |||||s2 |||| ||und|d |
| 245 10 - TITLE STATEMENT | |
| Title | Salt selection for basic drugs |
| 490 0# - SERIES STATEMENT | |
| Volume/sequential designation | International Journal of Pharmaceutics, 33(1-3), p.201-217, 1986 |
| 520 3# - SUMMARY, ETC. | |
| Summary, etc. | An attempt has been made using a Kepner-Tregoe decision analysis approach to provide rationale to salt selection for basic drugs. The selection objectives are reviewed in terms of the 'essential' (MUSTS)and 'desirable' (WANTS)issues. The desired characteristics of the salt form, given sufficient strength and toxicological suitability of the conjugate acid, are then discussed on the basis of the various pivotal physicochemical properties; melting point, aqueous solubility and dissolution rate, stability and hydrophobicity. Several trends are established which can then assist the decision of which range of salt forms to evaluate to overcome a particular problem with a basic drug. It is concluded that it is important to view the choice of salt form for development as a compromise, with particular focus on the correctly weighted desires to obtain the best balanced choice. |
| 650 14 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | SALT FORM SELECTION |
| 650 14 - SUBJECT ADDED ENTRY--TOPICAL TERM | |
| Topical term or geographic name entry element | PHARMACEUTICAL SALTS |
| 700 12 - ADDED ENTRY--PERSONAL NAME | |
| Personal name | Gould, P.L. |
| 856 40 - ELECTRONIC LOCATION AND ACCESS | |
| Uniform Resource Identifier | <a href="https://drive.google.com/file/d/1H3o0dNJTu2J6CBl7_FN8XtA4W396SL0d/view?usp=drivesdk">https://drive.google.com/file/d/1H3o0dNJTu2J6CBl7_FN8XtA4W396SL0d/view?usp=drivesdk</a> |
| Public note | Para ver el documento ingresa a Google con tu cuenta: @cicy.edu.mx |
| 942 ## - ADDED ENTRY ELEMENTS (KOHA) | |
| Source of classification or shelving scheme | Clasificación local |
| Koha item type | Documentos solicitados |
| Lost status | Source of classification or shelving scheme | Damaged status | Not for loan | Collection | Home library | Current library | Shelving location | Date acquired | Total checkouts | Full call number | Date last seen | Price effective from | Koha item type |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Clasificación local | Ref1 | CICY | CICY | Documento préstamo interbibliotecario | 25.06.2025 | B-14951 | 25.06.2025 | 25.06.2025 | Documentos solicitados |
