Verticilide, a new ryanodine-binding inhibitor, produced byVerticilliumsp. FKI-1033
Tipo de material:
TextoSeries ; The Journal of Antibiotics , 63(2), p.77-82, 2010Trabajos contenidos: - Kazuro Shiomi
- Ryosuke Matsui
- Atsuo Kakei
- Yuichi Yamaguchi
- Rokuro Masuma
- Hiroko Hatano
- Noriko Arai
- Noriko Arai
- Haruo Tanaka
- Susumu Kobayashi
- Andreas Turberg
- Satoshi Omura
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A new ryanodine-binding inhibitor, verticilide, was isolated from the cultured broth of a fungus,Verticilliumsp. FKI-1033. It is a 24-membered ring cyclic depsipeptide, its structure being elucidated as cyclo[(2R)-2-hydroxyheptanoyl-N-methyl-L-alanyl]4. Verticilide inhibited ryanodine binding to ryanodine receptors in the cockroach at an IC50value of 4.2lM, whereas inhibition against mouse ryanodine receptors was weak (IC50¼53.9lM).
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